Clinical Development

Our Pipeline

CSA-144, our lead Ceragenin compound, is being developed across multiple therapeutic areas with the potential to address significant unmet medical needs.

7
Active Programs
3
Therapeutic Areas
2
Formulations

Development Status

Current clinical development progress for all CSA-144 programs.

Therapeutic Area
Candidate
Indication/Target
Preclinical POC
Phase 1
Phase 2
Phase 3
Dermatology
CSA-144(Topical Hydrogel)
Diabetic Foot UlcersLead
CSA-144(Topical Hydrogel)
Epidermolysis Bullosa
CSA-144(Topical Cream)
Severe Atopic Dermatitis
CSA-144(Topical Cream)
Antiscarring Treatment
CSA-144(Topical Hydrogel)
Topical Antimicrobial
Women's Health
CSA-144(Topical Hydrogel)
STI Prevention
Antifungal
CSA-144(Topical Cream)
Onychomycosis
Dermatology
Women's Health
Antifungal

Program Details

In-depth information about each of our development programs.

CSA-144

Topical Hydrogel

Lead Program
DermatologyPhase 1

Diabetic Foot Ulcers

CSA-144 Topical Hydrogel for the treatment of diabetic foot ulcers, a chronic wound condition affecting millions of diabetic patients worldwide.

Unmet Need

Diabetic foot ulcers affect 15-25% of diabetics during their lifetime, with limited effective treatment options and high amputation rates.

Target Population

Approximately 537 million adults with diabetes globally, with 9.1-26.1 million developing foot ulcers annually.

Mechanism

Broad-spectrum antimicrobial activity prevents infection while promoting wound healing through biofilm disruption.

CSA-144

Topical Hydrogel

DermatologyPreclinical POC

Epidermolysis Bullosa

CSA-144 for Epidermolysis Bullosa, a rare genetic skin disorder causing fragile skin that blisters easily. Orphan drug designation.

Unmet Need

No FDA-approved treatments specifically for EB wound management. Patients face chronic wounds and high infection risk.

Target Population

Estimated 500,000 people worldwide affected by various forms of EB.

Mechanism

Antimicrobial protection for fragile skin wounds while being non-cytotoxic to healing tissue.

CSA-144

Topical Cream

DermatologyDiscovery

Severe Atopic Dermatitis

CSA-144 Topical Cream for severe atopic dermatitis patients with specific genetic markers indicating Ceragenin responsiveness.

Unmet Need

Atopic dermatitis affects up to 20% of children and 3% of adults, with severe cases requiring better treatment options.

Target Population

Patients with moderate-to-severe atopic dermatitis and identified genetic markers.

Mechanism

Reduces skin colonization by S. aureus, a key driver of AD flares and inflammation.

CSA-144

Topical Cream

DermatologyDiscovery

Antiscarring Treatment

CSA-144 Topical Cream developed to prevent and reduce scarring following surgical procedures or traumatic wounds.

Unmet Need

Significant scarring affects quality of life for millions of surgery and trauma patients annually.

Target Population

Post-surgical patients and individuals with healing traumatic wounds.

Mechanism

Modulates wound healing environment to reduce excessive collagen deposition and scar formation.

CSA-144

Topical Hydrogel

DermatologyDiscovery

Topical Antimicrobial

CSA-144 Topical Hydrogel as a broad-spectrum topical antimicrobial for various skin and wound infections.

Unmet Need

Rising antimicrobial resistance limits treatment options for common skin infections.

Target Population

Patients with bacterial, fungal, or mixed skin infections including drug-resistant strains.

Mechanism

Membrane-disrupting mechanism provides rapid, broad-spectrum activity without resistance development.

CSA-144

Topical Hydrogel

Women's HealthDiscovery

STI Prevention

CSA-144 Topical Hydrogel for the prevention of sexually transmitted infections through topical application.

Unmet Need

STIs continue to rise globally with limited prevention options beyond barrier methods.

Target Population

Adults seeking additional protection against common STIs.

Mechanism

Topical antimicrobial barrier provides protection against bacterial and viral pathogens.

CSA-144

Topical Cream

AntifungalDiscovery

Onychomycosis

CSA-144 Topical Cream for the treatment of onychomycosis (toenail fungus), a common fungal nail infection.

Unmet Need

Current topical treatments have low cure rates; oral antifungals carry systemic side effects.

Target Population

Estimated 10% of the general population affected by onychomycosis.

Mechanism

Penetrates nail bed to deliver potent antifungal activity directly to the site of infection.

Development Process

Our rigorous clinical development process ensures the safety and efficacy of our Ceragenin-based therapeutics.

Stage 1

Discovery

Identify and validate drug candidates through laboratory research and early testing.

  • Target identification
  • Lead compound optimization
  • In vitro efficacy studies
  • Initial safety assessment
Stage 2

Preclinical POC

Conduct comprehensive laboratory and animal studies to establish proof of concept.

  • Pharmacokinetic studies
  • Toxicology assessments
  • Formulation development
  • IND-enabling studies
Stage 3

Phase 1

First-in-human trials to evaluate safety, tolerability, and pharmacokinetics.

  • Safety and tolerability
  • Dose escalation studies
  • Pharmacokinetic profiling
  • Initial efficacy signals
Stage 4

Phase 2

Controlled trials to assess efficacy and optimal dosing in target patient population.

  • Efficacy evaluation
  • Dose-response studies
  • Safety monitoring
  • Endpoint validation
Stage 5

Phase 3

Large-scale pivotal trials to confirm safety and efficacy for regulatory approval.

  • Pivotal efficacy trials
  • Long-term safety data
  • Regulatory submissions
  • Commercialization prep

Clinical development timelines vary based on indication complexity, regulatory requirements, and trial enrollment. Our experienced team works to advance programs efficiently while maintaining the highest standards of patient safety.